Saturday
|
1:00 pm - 5:00 pm |
Arrival and Check-in
|
3:00 pm - 3:15 pm |
Introductory Comments by GRC Site Staff / Welcome from the GRS Chair
|
3:15 pm - 4:00 pm |
Keynote Session: Cyclic Nucleotide Phosphodiesterases: Potential Therapeutic Targets for Alcohol use Disorder
Discussion Leader: Ben Rombaut (University Hasselt, Belgium)
|
3:15 pm - 3:45 pm |
Hanting Zhang (Qingdao University School of Pharmacy, China)
"PDE, a Valve for the Control of Alcohol Drinking"
|
3:45 pm - 4:00 pm |
Discussion
|
4:00 pm - 5:30 pm |
Poster Session
|
5:30 pm - 7:30 pm |
Mapping the Pathway of Interactions to Investigate Functional Impact
Discussion Leaders: Romy Thomas (Max-Delbrück-Centrum for Molecular Medicine Berlin, Germany)
|
5:30 pm - 5:50 pm |
Introduction by Discussion Leader
|
5:50 pm - 6:05 pm |
Ben Rombaut (University Hasselt, Belgium)
"PDE4B as a Key Regulator of out of Control Microglia"
|
6:05 pm - 6:10 pm |
Discussion
|
6:10 pm - 6:25 pm |
Emma Parsons (University of Glasgow, United Kingdom)
"Analysis of Differentially Expressed Genes in PDE4D7 Silenced Prostate Cancer Cell Lines"
|
6:25 pm - 6:30 pm |
Discussion
|
6:30 pm - 6:45 pm |
Maria Ercu (Max-Delbrück-Centrum für Molekulare Medizin, Anchored Signalling department, Germany)
"Phosphodiesterase 3A Mutations Protect from Cardiac Damage"
|
6:45 pm - 6:50 pm |
Discussion
|
6:50 pm - 7:05 pm |
Nicolas Liem (Humboldt-University of Berlin, Germany)
"Novel Light-Activated Phosphodiesterases with High Affinity"
|
7:05 pm - 7:10 pm |
Discussion
|
7:10 pm - 7:25 pm |
Bernadin Ndongson Dongmo (University of Oslo, Norway)
"Effects of AAV9-Mediated Cardiac Phosphodiesterase 4B and 2A Overexpression in a Mouse Model of Heart Failure with Preserved Ejection Fraction"
|
7:25 pm - 7:30 pm |
Discussion
|
8:00 pm - 9:00 pm |
Dinner
|
Sunday
|
7:30 am - 8:30 am |
Breakfast
|
9:00 am - 11:00 am |
Recent Progress for Phosphodiesterases as Therapeutic Targets
Discussion Leader: Emma Parsons (University of Glasgow, United Kingdom)
|
9:00 am - 9:20 am |
Introduction by Discussion Leader
|
9:20 am - 9:35 am |
Elka Kyurkchieva (University of Glasgow, United Kingdom)
"Targeted Degradation of Short and Super-Short PDE4D Isoforms Using Bi-Functional Proteolysis Targeting Chimera (PROTAC) Molecules"
|
9:35 am - 9:40 am |
Discussion
|
9:40 am - 9:55 am |
Emily Willems (Maastricht University - School for Mental Health and Neuroscience, The Netherlands)
"Specific Inhibition of Phosphodiesterase 4D Long Isoforms Improves Neuronal Plasticity and Protects Against Aß Toxicity In Vitro"
|
9:55 am - 10:00 am |
Discussion
|
10:00 am - 10:15 am |
Chloe Gulliver (University of Glasgow, United Kingdom)
"PDE4D7 Expression Influences Prostate Cancer Development and Therapeutic Resistance."
|
10:15 am - 10:20 am |
Discussion
|
10:20 am - 10:35 am |
Ying Xu (Rutgers, The State University of New Jersey, United States)
"Phosphodiesterase Inhibitors and Alzheimer’s Disease: from Nature to Pharmacy"
|
10:35 am - 10:40 am |
Discussion
|
10:40 am - 10:55 am |
Walma Vasconcelos (Universite Paris Saclay, France)
"Regulation of Cardiac Pacemaker Activity by PDE4B and PDE4D"
|
10:55 am - 11:00 am |
Discussion
|
11:00 am - 12:30 pm |
Poster Session
Coffee will be served in the poster area from 11:00 am - 11:30 am
|
12:30 pm - 1:30 pm |
Lunch
|
1:30 pm - 2:30 pm |
Mentorship Component: Building Academic Resilience
Discussion Leader: Emily Willems (Maastricht University - School for Mental Health and Neuroscience, The Netherlands)
|
1:30 pm - 1:50 pm |
Leila Gobejishvili (University of Louisville, United States)
"Experiences from Our Own Careers"
|
1:50 pm - 2:00 pm |
Discussion
|
2:00 pm - 2:20 pm |
Tim Vanmierlo (Hasselt University / Maastricht University, Belgium)
"Experiences from Our Own Careers"
|
2:20 pm - 2:30 pm |
Discussion
|
2:30 pm - 3:00 pm |
Evaluation Period
Fill in GRS Evaluation Forms
|
3:00 pm |
Seminar Concludes
|