| SUNDAY | 
| 2:00 pm - 9:00 pm | Arrival and Check-in (Office Closed 6:00 pm - 7:00 pm) | 
| 5:00 pm - 6:00 pm | Welcome Mixer | 
| 6:00 pm | Dinner | 
| 7:30 pm - 7:40 pm | Welcome / Introductory Comments by GRC Site Staff and Conference Chair, Chris Moody | 
| 7:30 pm - 9:30 pm | NEW METHODOLOGY IN THE SYNTHESIS OF HETEROCYCLIC COMPOUNDS I | 
|  | Discussion Leader: J. Ramon Vargas (Eastman Kodak) | 
| 7:40 pm - 8:25 pm | Jeffrey Aubé (University of Kansas) "Heterocyclic libraries inspired by natural products and peptides"
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| 8:25 pm - 8:35 pm | Discussion | 
| 8:35 pm - 9:20 pm | Viresh Rawal (University of Chicago) "Recent progress on the total synthesis of indole alkaloids"
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| 9:15 pm - 9:30 pm | Discussion | 
| MONDAY | 
| 7:30 am - 8:30 am | Breakfast | 
| 9:00 am - 12:30 pm | CATALYSIS IN HETEROCYCLIC CHEMISTRY | 
|  | Discussion Leader: Julia M. Clay (Eli Lilly) | 
| 9:00 am - 9:50 am | Gregory C. Fu (Massachusetts Institute of Technology) "Palladium- and nickel-catalyzed coupling reactions"
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| 9:50 am - 10:00 am | Discussion | 
| 10:00 am | Coffee Break / Group Photo (10:15 am) | 
| 10:30 am - 11:00 am | Janis Louie (University of Utah) "Insights into Ni-catalyzed pyridine formation"
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| 11:00 am - 11:10 am | Discussion | 
| 11:10 am - 11:40 am | Tom G. Driver (University of Illinois at Chicago) "Transition metal-catalyzed reactions of azides"
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| 11:40 am - 11:50 am | Discussion | 
| 11:50 am - 12:20 pm | Helena Malinakova (University of Kansas) "Transition metal-catalyzed multi-component coupling reactions and reaction sequences for the synthesis of medicinally relevant heterocycles"
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| 12:20 pm - 12:30 pm | Discussion | 
| 12:30 pm | Lunch | 
| 1:30 pm - 4:00 pm | Free Time | 
| 4:00 pm - 6:00 pm | Poster Session 1 (Convenor: Ramon Vargas) | 
| 6:00 pm | Dinner | 
| 7:30 pm - 9:30 pm | SYNTHESIS OF HETEROCYCLIC NATURAL PRODUCTS | 
|  | Discussion Leader: Tom Pettus (UC Santa Barbara) | 
| 7:30 pm - 8:00 pm | Richmond Sarpong (University of California, Berkeley) "A unified strategy for the total synthesis of "miscellaneous" Lycopodium alkaloids"
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| 8:00 pm - 8:10 pm | Discussion | 
| 8:10 pm - 9:10 pm | Samuel J. Danishefsky (Columbia University/Sloan Kettering Institute) "Biologic level molecules through chemical synthesis"
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| 9:10 pm - 9:30 pm | Discussion | 
| TUESDAY | 
| 7:30 am - 8:30 am | Breakfast | 
| 9:00 am - 12:30 pm | NEW ROUTES TO BIOLOGICALLY ACTIVE HETEROCYCLES I | 
|  | Discussion Leader: Jon Njardarson (Cornell University) | 
| 9:00 am - 9:30 am | John Gilday (AstraZeneca) "Identification and development of manufacturing routes to the anilinoquinazoline, gefitinib, active ingredient of Iressa®"
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| 9:30 am - 9:35 am | Discussion | 
| 9:35 am - 10:20 am | Mercedes Álvarez (IRB, Barcelona) "Synthesis of polyheterocyclic nitrogen containing marine natural products"
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| 10:20 am - 10:30 am | Discussion | 
| 10:30 am | Coffee Break | 
| 11:00 am - 11:30 am | Kevin W. Gillman (Bristol Myers Squibb) "Heterocyclic gamma-secretase inhibitors for the treatment of Alzheimer’s disease"
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| 11:30 am - 11:35 am | Discussion | 
| 11:35 am - 12:20 pm | Louis Barriault (University of Ottawa) "Harvest in the pericyclic reaction garden"
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| 12:20 pm - 12:30 pm | Discussion | 
| 12:30 pm | Lunch | 
| 1:30 pm - 6:00 pm | Free Time | 
| 6:00 pm | Dinner | 
| 7:30 pm - 9:30 pm | HETEROCYCLIC NATURAL PRODUCTS AND THEIR BIOSYNTHESIS | 
|  | Discussion Leader: George Sheppard (Abbott) | 
| 7:30 pm - 8:00 pm | Sarah E. O’Connor (Massachusetts Institute of Technology) "Metabolic reprograming of alkaloid biosynthesis"
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| 8:00 pm - 8:05 pm | Discussion | 
| 8:05 pm - 8:25 pm | Craig A. Hutton (University of Melbourne) "Recent progress in the synthesis of cyclic peptide natural products"
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| 8:25 pm - 8:30 pm | Discussion | 
| 8:30 pm - 9:20 pm | Robert M. Williams (Colorado State University) "Total synthesis as a vehicle for penetrating biomechanistic puzzles: challenges in heterocyclic natural products chemistry"
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| 9:20 pm - 9:30 pm | Discussion | 
| WEDNESDAY | 
| 7:30 am - 8:30 am | Breakfast | 
| 9:00 am - 12:30 pm | NEW STRATEGIES TOWARDS HETEROCYCLIC COMPOUNDS | 
|  | Discussion Leader: H. Ila (Indian Institute of Technology, Kanpur) | 
| 9:00 am - 9:30 am | Anna Mapp (University of Michigan) "Small molecule transcriptional switches"
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| 9:30 am - 9:35 am | Discussion | 
| 9:35 am - 10:20 am | Thorsten Bach (Technische Universität, Munich) "Heterocycles in photochemical and organometallic reactions"
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| 10:20 am - 10:30 am | Discussion | 
| 10:30 am - 10:40 am | Business Meeting Part 1 | 
|  | (Nominations for the next Vice Chair) | 
| 10:40 am | Coffee Break | 
| 11:10 am - 11:30 am | Neil Garg (UCLA) "Studies in heterocycle synthesis: indoles, indolines, and indolynes"
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| 11:30 am - 11:35 am | Discussion | 
| 11:35 am - 12:20 pm | Donald Craig (Imperial College, London) "From aziridines to alkaloids: method development and total synthesis"
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| 12:20 pm - 12:30 pm | Discussion | 
| 12:30 pm | Lunch | 
| 1:30 pm - 4:00 pm | Free Time | 
| 4:00 pm - 6:00 pm | Poster Session 2 (Convenor: Ramon Vargas) | 
| 6:00 pm | Dinner | 
| 7:30 pm - 9:30 pm | NEW METHODOLOGY IN THE SYNTHESIS OF HETEROCYCLIC COMPOUNDS II | 
|  | Discussion Leader: Jennifer Love (University of British Columbia) | 
| 7:30 pm - 8:00 pm | Paul Vogt (SiGNa) "Application of stabilized alkali metals in heterocyclic synthesis"
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| 8:00 pm - 8:05 pm | Discussion | 
| 8:05 pm - 8:25 pm | James P. Stambuli (Ohio State University) "Nickel-catalyzed synthesis of oxazoles via C-S activation"
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| 8:25 pm - 8:30 pm | Discussion | 
| 8:30 pm - 9:20 pm | Sam Zard (École Polytechnique, Paris) "Adventures in radical chemistry: some unusual routes to heterocycles"
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| 9:20 pm - 9:30 pm | Discussion | 
| THURSDAY | 
| 7:30 am - 8:30 am | Breakfast | 
| 9:00 am - 12:30 pm | NEW ROUTES TO BIOLOGICALLY ACTIVE HETEROCYCLES II | 
|  | Discussion Leader: Dan Elbaum (FoldRx Pharmaceuticals) | 
| 9:00 am - 9:25 am | Brian Shook (Johnson & Johnson) "The design and Synthesis of indenopyrimidines as dual adenosine A2a/A1 antagonists for the treatment of Parkinson's disease"
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| 9:25 am - 9:30 am | Discussion | 
| 9:30 am - 9:55 am | R. Jason Herr (Albany Molecular Research Inc) "Small adventures in total synthesis"
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| 9:55 am - 10:00 am | Discussion | 
| 10:00 am - 10:30 am | Business Meeting Part 2 | 
|  | (Fill out Conference Evaluation Forms; Discuss future Site & Scheduling preferences; Election of the next Vice Chair) | 
| 10:30 am | Coffee Break | 
| 11:00 am - 11:30 am | Tehshik P. Yoon (University of Wisconsin, Madison) "Cycloadditions by visible light photocatalysis"
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| 11:30 am - 11:35 am | Discussion | 
| 11:35 am - 11:55 am | Amy Dounay (Pfizer Global R&D) "Design, synthesis, and pharmacological evaluation of phenoxy pyridyl derivatives as norepinephrine reuptake inhibitors and 5-HT1A partial agonists"
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| 11:55 am - 12:00 pm | Discussion | 
| 12:00 pm - 12:25 pm | Scott Coffey (Eli Lilly) "Process development of an NK-1 antagonist"
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| 12:25 pm - 12:30 pm | Discussion | 
| 12:30 pm | Lunch | 
| 1:30 pm - 6:00 pm | Free Time / Optional Wine Tasting Social (4:00 pm - 6:00 pm) | 
| 6:00 pm | Dinner | 
| 7:30 pm - 9:30 pm | PERSPECTIVES ON HETEROCYCLIC CHEMISTRY | 
|  | The challenges posed by the synthesis of complex heterocyclic compounds | 
|  | Discussion Leader: Chris Moody (University of Nottingham) | 
| 7:30 am - 8:15 pm | Jon Rainier (University of Utah) "Approaches to heterocycles at 4700 feet above sea level"
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| 8:15 pm - 8:20 pm | Discussion | 
| 8:20 pm - 9:05 pm | Stephen F. Martin (University of Texas, Austin) "Recent advances in the synthesis of complex heterocyclic natural products"
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| 9:05 pm - 9:15 pm | Discussion | 
| 9:15 pm - 9:30 pm | J. Ramon Vargas (Eastman Kodak) "Vice Chair’s Closing Remarks"
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| FRIDAY | 
| 7:30 am - 8:30 am | Breakfast | 
| 9:00 am | Departure |