Saturday 
 
 
2:00 pm - 5:00 pm 
	
Arrival and Check-in
 
 
						
3:30 pm - 3:45 pm 
	
Introductory Comments by GRC Site Staff / Welcome from the GRS Chair
 
 
						
3:45 pm - 4:30 pm 
	
Keynote Session: Clinical Significance / Pharmacological Impact 
 
 
 
						
3:45 pm - 4:05 pm 
	
"Clinical Significance of Multidrug Efflux Pumps: From Biology to Cancer Therapies" 
 
 
 
						
4:05 pm - 4:10 pm 
	
Discussion
 
 
						
4:10 pm - 4:25 pm 
	
"Targeting HIV Reservoirs in Brain by Inhibition of P-Glycoprotein at
the Blood-Brain Barrier" 
 
 
 
						
4:25 pm - 4:30 pm 
	
Discussion
 
 
						
4:30 pm - 6:00 pm 
	
Poster Session 
 
 
						
6:00 pm - 7:00 pm 
	
Dinner
 
 
						
7:30 pm - 9:30 pm 
	
Application to Drug Discovery 
 
 
 
						
7:30 pm - 7:45 pm 
	
"Biophysical Characterizations of Drug Binding Coupled to ATP Hydrolysis by P-Glycoprotein Reconstituted in Lipid Nanodiscs" 
 
 
 
						
7:45 pm - 7:50 pm 
	
Discussion
 
 
						
7:50 pm - 8:05 pm 
	
"Combination Therapy to Overcome ABC Transport Mediated Chemoresistance in a Colorectal Cancer Mouse Xenograft Model" 
 
 
 
						
8:05 pm - 8:10 pm 
	
Discussion
 
 
						
8:10 pm - 8:25 pm 
	
"Overcoming P-Glycoprotein-Associated Resistance in Chronic
Myelogenous Leukemia with Dasatinib-Based Prodrugs" 
 
 
 
						
8:25 pm - 8:30 pm 
	
Discussion
 
 
						
8:30 pm - 8:45 pm 
	
"Activity of the Dietary Flavonoid, Apigenin, Against Multidrug-Resistant Tumor Cells as Determined by Pharmacogenomics and Molecular Docking" 
 
 
 
						
8:45 pm - 8:50 pm 
	
Discussion
 
 
						
8:50 pm - 9:05 pm 
	
"Phenothiazines Against Antibiotic Resistance: Impact on Efflux Pumps Expression of B. pseudomallei " 
 
 
 
						
9:05 pm - 9:10 pm 
	
Discussion
 
 
						
9:10 pm - 9:25 pm 
	
"Efflux Pumps as Tools to Increase Biofuel Tolerance in Bacteria" 
 
 
 
						
9:25 pm - 9:30 pm 
	
Discussion
 
 
						
	Sunday 
 
 
7:30 am - 8:30 am 
	
Breakfast
 
 
						
9:00 am - 11:00 am 
	
Keynote Session: Biochemical Studies / Omics Approaches 
 
 
 
						
9:00 am - 9:20 am 
	
"Deciphering the Molecular Details of Substrate Transport and Energy Coupling in Bacterial Multidrug Efflux Pumps" 
 
 
 
						
9:20 am - 9:25 am 
	
Discussion
 
 
						
9:25 am - 9:40 am 
	
"Hoechst 33342 Is a Hidden 'Janus' Amongst Substrates for the Multidrug Efflux Pump LmrP" 
 
 
 
						
9:40 am - 9:45 am 
	
Discussion
 
 
						
9:45 am - 10:00 am 
	
"Transcriptional Activation of Genes Encoding the MacAB Macrolide Efflux Pump by MisR in Neisseria gonorrhoeae " 
 
 
 
						
10:00 am - 10:05 am 
	
Discussion
 
 
						
10:05 am - 10:20 am 
	
"Carbonyl Stress Induces the Efflux System MexEF-OprN in Pseudomonas aeruginosa  via a Novel Transcriptional Regulator, CmrA" 
 
 
 
						
10:20 am - 10:25 am 
	
Discussion
 
 
						
10:25 am - 10:40 am 
	
"Genomic and Transcriptomic Profiling of Resistant CEM/ADR-5000 and Sensitive CCRF-CEM Leukaemia Cells for Unravelling the Full Complexity of Multi-Factorial Multidrug Resistance" 
 
 
 
						
10:40 am - 10:45 am 
	
Discussion
 
 
						
10:45 am - 11:00 am 
	
General Discussion
 
 
						
11:00 am - 12:30 pm 
	
Poster Session 
Coffee will be served in the poster area from 11:00 am - 11:30 am 
 
 
						
12:30 pm - 1:30 pm 
	
Lunch
 
 
						
1:30 pm - 2:30 pm 
	
Mentorship Component: Career Development Panel 
 
 
 
						
1:30 pm - 2:30 pm 
	
Panel Discussion 
Career Development Panel 
 
 
 
						
2:30 pm - 3:00 pm 
	
Evaluation Period 
Fill in GRS Evaluation Forms 
 
 
						
3:00 pm 
	
Seminar Concludes