Sunday 
 
 
2:00 pm - 9:00 pm 
	
Arrival and Check-in
 
 
						 
						 
					
						
						
6:00 pm - 7:00 pm 
	
Dinner
 
 
						 
						 
					
						
						
7:30 pm - 7:40 pm 
	
Introductory Comments by GRC Site Staff / Welcome from the GRC Chair
 
 
						 
						 
					
						
						
7:40 pm - 9:30 pm 
	
Stereochemical and Atomic Control in Organic Synthesis 
 
 
 
						 
						 
					
						
						
7:40 pm - 8:10 pm 
	
"Copper-Catalyzed Aminofunctionalization of Alkenes and Dienes" 
 
 
 
						 
						 
					
						
						
8:10 pm - 8:15 pm 
	
Discussion
 
 
						 
						 
					
						
						
8:15 pm - 8:45 pm 
	
"Polarity Inversion Catalysis by the Conjugate Addition of Lewis Bases" 
 
 
 
						 
						 
					
						
						
8:45 pm - 8:50 pm 
	
Discussion
 
 
						 
						 
					
						
						
8:50 pm - 9:25 pm 
	
"Stereoselective Synthesis in Stereochemically Fluxional Systems" 
 
 
 
						 
						 
					
						
						
9:25 pm - 9:30 pm 
	
Discussion
 
 
						 
						 
					
						
						
	Monday 
 
 
7:30 am - 8:30 am 
	
Breakfast
 
 
						 
						 
					
						
						
9:00 am - 12:30 pm 
	
Installation and Uses of Halogens 
 
 
 
						 
						 
					
						
						
9:00 am - 9:30 am 
	
"Design and Development of a Convergent Synthesis of an Aminoquinoline NLRP3 Agonist" 
 
 
 
						 
						 
					
						
						
9:30 am - 9:35 am 
	
Discussion
 
 
						 
						 
					
						
						
9:35 am - 10:05 am 
	
"Development of a Palladium-Catalyzed Aryl Amidation for API Synthesis" 
 
 
 
						 
						 
					
						
						
10:05 am - 10:10 am 
	
Discussion
 
 
						 
						 
					
						
						
10:10 am - 10:35 am 
	
Coffee Break
 
 
						 
						 
					
						
						
10:35 am - 11:05 am 
	
"Technology Solutions to Unlock Access to Challenging Reactions on Scale" 
 
 
 
						 
						 
					
						
						
11:05 am - 11:10 am 
	
Discussion
 
 
						 
						 
					
						
						
11:10 am - 11:45 am 
	
"Teaching an Old Dog New Tricks: Selenium as a Catalyst for C-H Amination Reactions" 
 
 
 
						 
						 
					
						
						
11:45 am - 11:50 am 
	
Discussion
 
 
						 
						 
					
						
						
11:50 am - 12:25 pm 
	
"Late-Stage Functionalizations" 
 
 
 
						 
						 
					
						
						
12:25 pm - 12:30 pm 
	
Discussion
 
 
						 
						 
					
						
						
12:30 pm - 1:30 pm 
	
Lunch
 
 
						 
						 
					
						
						
1:30 pm - 4:00 pm 
	
Free Time
 
 
						 
						 
					
						
						
4:00 pm - 6:00 pm 
	
Poster Session 
 
 
						 
						 
					
						
						
6:00 pm - 7:00 pm 
	
Dinner
 
 
						 
						 
					
						
						
7:30 pm - 9:30 pm 
	
Innovative Strategies in C-C Bond Formation 
 
 
 
						 
						 
					
						
						
7:30 pm - 8:05 pm 
	
"En-Light-Ening C–H Functionalization" 
 
 
 
						 
						 
					
						
						
8:05 pm - 8:10 pm 
	
Discussion
 
 
						 
						 
					
						
						
8:10 pm - 8:45 pm 
	
"Site Selective Synthesis of Benzylic Collidinium Salts via Electrochemical C–H Functionalization" 
 
 
 
						 
						 
					
						
						
8:45 pm - 8:50 pm 
	
Discussion
 
 
						 
						 
					
						
						
8:50 pm - 9:25 pm 
	
"Alkyne Functionalization for Use in Organic Synthesis" 
 
 
 
						 
						 
					
						
						
9:25 pm - 9:30 pm 
	
Discussion
 
 
						 
						 
					
						
						
	Tuesday 
 
 
7:30 am - 8:30 am 
	
Breakfast
 
 
						 
						 
					
						
						
9:00 am - 12:30 pm 
	
 
 
						 
						 
					
						
						
9:00 am - 9:30 am 
	
"Process Development of Paxlovid: Milligrams to Metric Tons in 18 Months" 
 
 
 
						 
						 
					
						
						
9:30 am - 9:35 am 
	
Discussion
 
 
						 
						 
					
						
						
9:35 am - 10:05 am 
	
"Efficient Manufacturing Process for the Selective Estrogen Receptor Degrader GDC-9545 (Giredestrant)" 
 
 
 
						 
						 
					
						
						
10:05 am - 10:10 am 
	
Discussion
 
 
						 
						 
					
						
						
10:10 am - 10:35 am 
	
Coffee Break
 
 
						 
						 
					
						
						
10:35 am - 11:05 am 
	
"How a Crystallization Induced Dynamic Resolution Made Lenacapavir Possible" 
 
 
 
						 
						 
					
						
						
11:05 am - 11:10 am 
	
Discussion
 
 
						 
						 
					
						
						
11:10 am - 11:45 am 
	
"Catalysis with Foldamers" 
 
 
 
						 
						 
					
						
						
11:45 am - 11:50 am 
	
Discussion
 
 
						 
						 
					
						
						
11:50 am - 12:25 pm 
	
"High-Throughput Enantiopurity Analysis using Enantiomeric DNA-Based Sensors" 
 
 
 
						 
						 
					
						
						
12:25 pm - 12:30 pm 
	
Discussion
 
 
						 
						 
					
						
						
12:30 pm - 1:30 pm 
	
Lunch
 
 
						 
						 
					
						
						
1:30 pm - 4:00 pm 
	
Free Time
 
 
						 
						 
					
						
						
4:00 pm - 6:00 pm 
	
Poster Session 
 
 
						 
						 
					
						
						
6:00 pm - 7:00 pm 
	
Dinner
 
 
						 
						 
					
						
						
7:30 pm - 9:30 pm 
	
Behold the Power of Light 
 
 
 
						 
						 
					
						
						
7:30 pm - 8:05 pm 
	
"New Avenues in Synthesis via Organic Photoredox Catalysis" 
 
 
 
						 
						 
					
						
						
8:05 pm - 8:10 pm 
	
Discussion
 
 
						 
						 
					
						
						
8:10 pm - 8:45 pm 
	
"Recreation by Umpolung: Amide and Peptide Synthesis" 
 
 
 
						 
						 
					
						
						
8:45 pm - 8:50 pm 
	
Discussion
 
 
						 
						 
					
						
						
8:50 pm - 9:25 pm 
	
"Electrophylic Deborylations in Synthesis" 
 
 
 
						 
						 
					
						
						
9:25 pm - 9:30 pm 
	
Discussion
 
 
						 
						 
					
						
						
	Wednesday 
 
 
7:30 am - 8:30 am 
	
Breakfast
 
 
						 
						 
					
						
						
8:30 am - 9:00 am 
	
Group Photo
 
 
						 
						 
					
						
						
9:00 am - 12:30 pm 
	
More C-C Bond Formation and Methods 
 
 
 
						 
						 
					
						
						
9:00 am - 9:25 am 
	
"Evolution of Adagrasib’s Commercial Manufacturing Route" 
 
 
 
						 
						 
					
						
						
9:25 am - 9:35 am 
	
Discussion
 
 
						 
						 
					
						
						
9:35 am - 10:00 am 
	
"Converting a Biorenewable Solvent into an Active Pharmaceutical Ingredient" 
 
 
 
						 
						 
					
						
						
10:00 am - 10:10 am 
	
Discussion
 
 
						 
						 
					
						
						
10:10 am - 10:35 am 
	
Coffee Break
 
 
						 
						 
					
						
						
10:35 am - 11:00 am 
	
"Hybrid Pd-Radical Chemistry: New Mechanism, New Possibilities" 
 
 
 
						 
						 
					
						
						
11:00 am - 11:10 am 
	
Discussion
 
 
						 
						 
					
						
						
11:10 am - 11:35 am 
	
"Enantioselective Chemical Synthesis Methods via Cooperative Catalysis" 
 
 
 
						 
						 
					
						
						
11:35 am - 11:45 am 
	
Discussion
 
 
						 
						 
					
						
						
11:45 am - 12:10 pm 
	
"Synthesis of Neuroprotective Limonoid Natural Products" 
 
 
 
						 
						 
					
						
						
12:10 pm - 12:20 pm 
	
Discussion
 
 
						 
						 
					
						
						
12:20 pm - 12:30 pm 
	
General Discussion
 
 
						 
						 
					
						
						
12:30 pm - 1:30 pm 
	
Lunch
 
 
						 
						 
					
						
						
1:30 pm - 4:00 pm 
	
Free Time
 
 
						 
						 
					
						
						
4:00 pm - 6:00 pm 
	
Poster Session 
 
 
						 
						 
					
						
						
6:00 pm - 7:00 pm 
	
Dinner
 
 
						 
						 
					
						
						
7:00 pm - 7:30 pm 
	
Business Meeting 
Nominations for the Next Vice Chair(s); Complete the GRC Evaluation Forms; Discuss Future Dates and Venue; Election of the Next Vice Chair(s) 
 
 
						 
						 
					
						
						
7:30 pm - 9:30 pm 
	
 
 
						 
						 
					
						
						
7:30 pm - 8:05 pm 
	
"Understanding, Improving and Controlling Processes by Realtime HPLC" 
 
 
 
						 
						 
					
						
						
8:05 pm - 8:10 pm 
	
Discussion
 
 
						 
						 
					
						
						
8:10 pm - 8:45 pm 
	
"Mapping Catalytic Oxidative Decarboxylative Coupling Reactions" 
 
 
 
						 
						 
					
						
						
8:45 pm - 8:50 pm 
	
Discussion
 
 
						 
						 
					
						
						
8:50 pm - 9:25 pm 
	
"Synthesis Design through the Lens of Flow Chemistry" 
 
 
 
						 
						 
					
						
						
9:25 pm - 9:30 pm 
	
Discussion
 
 
						 
						 
					
						
						
	Thursday 
 
 
7:30 am - 8:30 am 
	
Breakfast
 
 
						 
						 
					
						
						
9:00 am - 12:30 pm 
	
 
 
						 
						 
					
						
						
9:00 am - 9:35 am 
	
"Unraveling the Mechanism of Electron Transfer from Samarium(II)-Proton Donor Complexes." 
 
 
 
						 
						 
					
						
						
9:35 am - 9:40 am 
	
Discussion
 
 
						 
						 
					
						
						
9:40 am - 10:15 am 
	
"Adventures in Flow Chemistry – Towards Continuous Manufacturing of APIs" 
 
 
 
						 
						 
					
						
						
10:15 am - 10:20 am 
	
Discussion
 
 
						 
						 
					
						
						
10:20 am - 10:40 am 
	
Coffee Break
 
 
						 
						 
					
						
						
10:40 am - 11:10 am 
	
"Accelerating Process Development with Automated Continuous Reactions and Online LC" 
 
 
 
						 
						 
					
						
						
11:10 am - 11:15 am 
	
Discussion
 
 
						 
						 
					
						
						
11:15 am - 11:35 am 
	
Short Talk Selected from Poster Abstracts
 
 
						 
						 
					
						
						
11:35 am - 11:40 am 
	
Discussion
 
 
						 
						 
					
						
						
11:40 am - 12:00 pm 
	
Short Talk Selected from Poster Abstracts
 
 
						 
						 
					
						
						
12:00 pm - 12:05 pm 
	
Discussion
 
 
						 
						 
					
						
						
12:05 pm - 12:25 pm 
	
Short Talk Selected from Poster Abstracts
 
 
						 
						 
					
						
						
12:25 pm - 12:30 pm 
	
Discussion
 
 
						 
						 
					
						
						
12:30 pm - 1:30 pm 
	
Lunch
 
 
						 
						 
					
						
						
1:30 pm - 4:00 pm 
	
Free Time
 
 
						 
						 
					
						
						
4:00 pm - 6:00 pm 
	
Poster Session 
 
 
						 
						 
					
						
						
6:00 pm - 7:00 pm 
	
Dinner
 
 
						 
						 
					
						
						
7:30 pm - 9:30 pm 
	
Chemistry on Complex Molecules 
 
 
 
						 
						 
					
						
						
7:30 pm - 8:05 pm 
	
"The Use of Natural-Abundance Stable Isotopes in Process Understanding - From Analysis to Synthesis" 
 
 
 
						 
						 
					
						
						
8:05 pm - 8:10 pm 
	
Discussion
 
 
						 
						 
					
						
						
8:10 pm - 8:45 pm 
	
"New Catalysts and Concepts for C-C and C-Heteroatom Bond Formation" 
 
 
 
						 
						 
					
						
						
8:45 pm - 8:50 pm 
	
Discussion
 
 
						 
						 
					
						
						
8:50 pm - 9:25 pm 
	
"Catalyst Speciation Controls Alkene Functionalization Pathways" 
 
 
 
						 
						 
					
						
						
9:25 pm - 9:30 pm 
	
Discussion
 
 
						 
						 
					
						
						
	Friday 
 
 
7:30 am - 8:30 am 
	
Breakfast
 
 
						 
						 
					
						
						
9:00 am 
	
Departure