Sunday
2:00 pm - 9:00 pm
Arrival and Check-in
6:00 pm - 7:00 pm
Dinner
7:30 pm - 7:40 pm
Introductory Comments by GRC Site Staff / Welcome from the GRC Chair
7:40 pm - 9:30 pm
Inorganic Nanomaterials in Medicine
7:40 pm - 7:45 pm
Introduction by Discussion Leader
7:45 pm - 8:10 pm
"Engineered-Surface Metal-Organic Frameworks as Drug Nanocarriers"
8:10 pm - 8:20 pm
Discussion
8:20 pm - 8:45 pm
"Bioorthogonal Catalysis Using Nanoparticle-Embedded Transition Metal Catalysts for Therapeutics and Diagnostics"
8:45 pm - 8:55 pm
Discussion
8:55 pm - 9:20 pm
"Autophagic Silicon Nanoparticles for Targeted Delivery of Therapeutics"
9:20 pm - 9:30 pm
Discussion
Monday
7:30 am - 8:30 am
Breakfast
9:00 am - 12:30 pm
Metal Homeostasis in Health and Disease
9:00 am - 9:05 am
Introduction by Discussion Leader
9:05 am - 9:35 am
"Inhibiting Metal-Mediated Demethylation to Reshape Cancer Epigenetics"
9:35 am - 9:50 am
Discussion
9:50 am - 10:20 am
"Siderophores and Their Potential Applications as Antimicrobials"
10:20 am - 10:30 am
Discussion
10:30 am - 11:00 am
Coffee Break
11:00 am - 11:30 am
"Potentiation of Oncolytic Virotherapy by Vanadium Compounds"
11:30 am - 11:45 am
Discussion
11:45 am - 12:15 pm
"Reprogramming the Chemical Reactivity of Metals in Cancer"
12:15 pm - 12:30 pm
Discussion
12:30 pm - 1:30 pm
Lunch
1:30 pm - 4:00 pm
Free Time
4:00 pm - 6:00 pm
Poster Session
6:00 pm - 7:00 pm
Dinner
7:30 pm - 9:30 pm
7:30 pm - 7:35 pm
Introduction by Discussion Leader
7:35 pm - 8:05 pm
"Ushering in the Digital Drug Design Revolution with Spherical Nucleic Acid Nanoparticle Conjugates"
8:05 pm - 8:15 pm
Discussion
8:15 pm - 8:45 pm
"Forge Therapeutics: Bioinorganic Directed Drug Discovery"
8:45 pm - 8:55 pm
Discussion
8:55 pm - 9:25 pm
"From Discovery to Company Formation: Views from a Venture Capital Investor"
9:25 pm - 9:30 pm
Discussion
Tuesday
7:30 am - 8:30 am
Breakfast
8:30 am - 9:00 am
Group Photo
9:00 am - 12:30 pm
Recent Developments in Metallodrugs
9:00 am - 9:05 am
Introduction by Discussion Leader
9:05 am - 9:35 am
"Gadolium Texaphyrins, Platinum and Gold"
9:35 am - 9:50 am
Discussion
9:50 am - 10:20 am
"Copper Complexes as Anticancer Agents: New Mechanistic Insights"
10:20 am - 10:30 am
Discussion
10:30 am - 11:00 am
Coffee Break
11:00 am - 11:30 am
"A Metal-Containing Drug Repurposed for Neglected Tropical Diseases"
11:30 am - 11:45 am
Discussion
11:45 am - 12:15 pm
"Innovative Metallo-Prodrug Strategies Leading to Multimodal Cancer Therapeutics"
12:15 pm - 12:30 pm
Discussion
12:30 pm - 1:30 pm
Lunch
1:30 pm - 4:00 pm
Free Time
4:00 pm - 6:00 pm
Poster Session
6:00 pm - 7:00 pm
Dinner
7:30 pm - 9:30 pm
7:30 pm - 7:35 pm
Introduction by Discussion Leader
7:35 pm - 8:05 pm
"Using Synthetic Heparan Sulfate to Treat Acute Liver Injury"
8:05 pm - 8:15 pm
Discussion
8:15 pm - 8:45 pm
"Manganese and Glycosaminoglycans in Tumor Progression: From Cell Migration to Premetastatic Niche Formation"
8:45 pm - 8:55 pm
Discussion
8:55 pm - 9:25 pm
"Glycans as Ligands in Bioinorganic Chemistry. Chemical and Biological Studies in Metalloglycomics"
9:25 pm - 9:30 pm
Discussion
Wednesday
7:30 am - 8:30 am
Breakfast
9:00 am - 12:30 pm
New Agents for Imaging Applications
9:00 am - 9:05 am
Introduction by Discussion Leader
9:05 am - 9:35 am
"Technetium and Rhenium Complexes with Aromatic Hydrocarbons as π-Ligands: An Entry into Biomimetic Imaging"
9:35 am - 9:50 am
Discussion
9:50 am - 10:20 am
"How Chelator Choice Impacts Biodistribution of Radiometal-Labeled Biomolecules"
10:20 am - 10:30 am
Discussion
10:30 am - 11:00 am
Coffee Break
11:00 am - 11:30 am
"From Cell Imaging to Predrug: The Renaissance of Metallosalens in Biological Applications"
11:30 am - 11:40 am
Discussion
11:40 am - 11:55 am
"Cutting Edge Fluorescence Imaging Strategies for Precise Regulation of Cellular Functions and Localized Theranostics"
11:55 am - 12:00 pm
Discussion
12:00 pm - 12:30 pm
Poster Previews
12:30 pm - 1:30 pm
Lunch
1:30 pm - 4:00 pm
Free Time
4:00 pm - 6:00 pm
Poster Session
6:00 pm - 7:00 pm
Dinner
7:00 pm - 7:30 pm
Business Meeting
Nominations for the Next Vice Chair; Fill in Conference Evaluation Forms; Discuss Future Site and Scheduling Preferences; Election of the Next Vice Chair
7:30 pm - 9:30 pm
Case Studies in Translational Research
7:30 pm - 7:35 pm
Introduction by Discussion Leader
7:35 pm - 8:05 pm
"Once upon a Time in Vienna: A Story from Ruthenium to Platinum"
8:05 pm - 8:15 pm
Discussion
8:15 pm - 8:45 pm
"Once upon a Time in Vienna: The Power of Activation by Reduction"
8:45 pm - 8:50 pm
Discussion
8:50 pm - 9:20 pm
"Once upon a Time in Vienna: Tumor-Specific Accumulation of Metallodrugs"
9:20 pm - 9:30 pm
Discussion
Thursday
7:30 am - 8:30 am
Breakfast
9:00 am - 12:30 pm
Analytical Techniques for Metals in Biological Systems
9:00 am - 9:05 am
Introduction by Discussion Leader
9:05 am - 9:35 am
"Methods for Comprehensive Analysis of Platinum Targets in Yeast and Mammalian Cancer Cells"
9:35 am - 9:50 am
Discussion
9:50 am - 10:20 am
"Metal Speciation in In Vitro and In Vivo Biological Activities from Drugs to Toxins"
10:20 am - 10:30 am
Discussion
10:30 am - 11:00 am
Coffee Break
11:00 am - 11:30 am
"Global Approaches to Metal Speciation: Metallomics"
11:30 am - 11:40 am
Discussion
11:40 am - 11:55 am
"Emerging Proteomics Methods to Elucidate Metallodrugs' Mechanisms of Action in the Cellular Context"
11:55 am - 12:00 pm
Discussion
12:00 pm - 12:30 pm
Poster Previews
12:30 pm - 1:30 pm
Lunch
1:30 pm - 4:00 pm
Free Time
4:00 pm - 6:00 pm
Poster Session
6:00 pm - 7:00 pm
Dinner
7:30 pm - 9:30 pm
Young Investigator Presentations
7:30 pm - 7:35 pm
Introduction by Discussion Leader
7:35 pm - 7:55 pm
"Therapeutic SIMCats: In Pursuit of Catalytic Medicines"
7:55 pm - 8:05 pm
Discussion
8:05 pm - 8:25 pm
"Metal-Chelating Antibiotics and Natural Products"
8:25 pm - 8:35 pm
Discussion
8:35 pm - 8:55 pm
"A Small Molecule that Transports Iron Promotes Iron Absorption and Hemoglobinization"
8:55 pm - 9:05 pm
Discussion
9:05 pm - 9:25 pm
"Rhenium(I) Complexes as Anticancer Agents: Challenges and Opportunities"
9:25 pm - 9:30 pm
Discussion
Friday
7:30 am - 8:30 am
Breakfast
9:00 am
Departure